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BPC-157's regulatory status is complex and may vary by use, jurisdiction, and product category, including FDA regulatory and safety concerns regarding certain BPC-157-related bulk substances used in compounding contexts

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Some have randomized controlled trials

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It has been demonstrated to induce mitochondrial damage and both intrinsic apoptotic and mPTP-driven cell death 13,14,15,16 via signalling pathways, indicating that its mode of action may involve BAX and BAK1

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