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DPP-4 inhibition extends this half-life and increases circulating active GLP-1 by approximately 2- to 3-fold, which is sufficient to engage high-density pancreatic islet receptors and produce glucose-dependent insulin secretion and glucagon suppression

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Orally administered semaglutide versus GLP-1 RAs in patients with type 2 diabetes previously receiving 12 oral antidiabetics: systematic review and network meta-analysis

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