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Lee HY, Suciu RM, Horning BD, Vinogradova EV, Ulanovskaya OA, Cravatt BF (2018) Covalent inhibitors of nicotinamide N-methyltransferase (NNMT) provide evidence for target engagement challenges in situ

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Levels of DIO2 mRNA and protein were markedly upregulated in OA cartilage 101