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Description
doi: 10.2174/138161209787185788

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Selectivity of NNMT inhibitors Test compounds were screened in biochemical assays for activity against three structurally similar methyltransferases, including catechol-O-methyltransferase (COMT), DNA (cytosine-5)-methyltransferase 1 (DNMT1), and protein arginine methyltransferase 3 (PRMT3)

That is 6,000 mcg per day of a peptide that saturates receptors at 100 mcg
